MRT68921 HCl
CAS No. 2070014-87-6
MRT68921 HCl ( —— )
Catalog No. M20090 CAS No. 2070014-87-6
MRT68921 hydrochloride is a potent inhibitor of both ULK1 and ULK2 (IC50s: 2.9 and 1.1 nM respectively).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 54 | In Stock |
|
10MG | 86 | In Stock |
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25MG | 178 | In Stock |
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50MG | 322 | In Stock |
|
100MG | 401 | In Stock |
|
200MG | Get Quote | In Stock |
|
500MG | Get Quote | In Stock |
|
1G | Get Quote | In Stock |
|
Biological Information
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Product NameMRT68921 HCl
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NoteResearch use only not for human use.
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Brief DescriptionMRT68921 hydrochloride is a potent inhibitor of both ULK1 and ULK2 (IC50s: 2.9 and 1.1 nM respectively).
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DescriptionMRT68921 hydrochloride is a potent inhibitor of both ULK1 and ULK2 (IC50s: 2.9 and 1.1 nM respectively).
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Synonyms——
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PathwayAutophagy
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TargetAutophagy
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RecptorULK1; ULK2
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Research Area——
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Indication——
Chemical Information
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CAS Number2070014-87-6
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Formula Weight471.04
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Molecular FormulaC25H34N6O·HCl
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Purity>98% (HPLC)
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SolubilityDMSO: 10 mg/mL;Water: 10 mg/mL
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SMILESCl.CN1CCc2cc(Nc3ncc(C4CC4)c(NCCCNC(=O)C4CCC4)n3)ccc2C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Petherick KJ et al. Pharmacological inhibition of ULK1 kinase blocks mammalian target of rapamycin (mTOR)-dependent autophagy. J Biol Chem. 2015 May 1;290(18):11376-83.
molnova catalog
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